SCHEMBL7606019

SCHEMBL7606019

CN(C)CC1=C(c2cccc(O)c2)c2cccc(Cl)c2OC1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 2/20 0.35
PTGS2 P35354 1/20 0.35
PIK3CA P42336 1/20 0.32
HSD17B1 P14061 4/20 0.32
HSD17B2 P37059 4/20 0.32
PGR P06401 1/20 0.32
AOC3 Q16853 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PRF1 P14222 1/20 0.31
KDR P35968 1/20 0.31
STK10 O94804 1/20 0.31
GSK3B P49841 1/20 0.31
SLK Q9H2G2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8006771 0.99 OPRD1 (0.35) OPRD1PTGS2PIK3CAHSD17B1HSD17B2
SCHEMBL7610280 0.82 PTGS2 (0.37) PTGS2HSD17B1HSD17B2MAPT
Hydrochloric Acid SCHEMBL8018678 0.81 ALDH1A1 (0.38) PTGS2PIK3CAHSD17B1HSD17B2MAPT
SCHEMBL7610149 0.81 CTNNB1 (0.33) OPRD1PTGS2PIK3CAHSD17B1HSD17B2
Hydrochloric Acid SCHEMBL8018169 0.80 PTGS2 (0.33) OPRD1PTGS2PIK3CAHSD17B1HSD17B2
SCHEMBL7611830 0.76 OPRD1 (0.35) OPRD1PTGS2PIK3CAHSD17B1HSD17B2
Hydrochloric Acid SCHEMBL8019741 0.75 OPRD1 (0.34) OPRD1PTGS2PIK3CAHSD17B1HSD17B2
SCHEMBL7611357 0.74 HTR7 (0.42) OPRD1HSD17B1HSD17B2MAPT
SCHEMBL7605210 0.74 ESR1 (0.44) PIK3CA
Hydrochloric Acid SCHEMBL8026792 0.73 HTR7 (0.41) OPRD1HSD17B1HSD17B2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922703-B1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds GRUENENTHAL GMBH (DE) 2002-12-04 EP disclosed
EP-0922703-A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds Grünenthal GmbH (DE) 1999-06-16 EP disclosed