SCHEMBL7610280

SCHEMBL7610280

CN(C)CC1=C(c2cccc(O)c2)c2ccccc2OC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.37
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 3/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HTR2B P41595 4/20 0.36
ADRA2A P08913 4/20 0.36
ADRA2B P18089 4/20 0.36
ADRA2C P18825 4/20 0.36
HRH1 P35367 3/20 0.36
KCNH2 Q12809 2/20 0.36
TSHR P16473 2/20 0.36
SLC22A1 O15245 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
HTR1A P08908 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8018678 0.99 ALDH1A1 (0.38) PTGS2ALDH1A1KDM4EMAPTRAB9A
SCHEMBL7605210 0.89 ESR1 (0.44) ESR1ESR2
Hydrochloric Acid SCHEMBL8016570 0.88 ESR1 (0.43) ESR1ESR2
SCHEMBL7605957 0.83 ESR1 (0.52) ALDH1A1KDM4EMAPTRAB9AGAA
SCHEMBL7606019 0.82 OPRD1 (0.35) PTGS2MAPTHSD17B1HSD17B2
Hydrochloric Acid SCHEMBL8006771 0.81 OPRD1 (0.35) PTGS2MAPTHSD17B1HSD17B2
SCHEMBL7591741 0.81 MTNR1A (0.44) ALDH1A1KDM4EMAPTHTR2BADRA2A
SCHEMBL7582908 0.81 CHRM2 (0.41) ALDH1A1KDM4EADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL8010759 0.80 MTNR1A (0.43) ALDH1A1KDM4EMAPTHTR2BADRA2A
Hydrochloric Acid SCHEMBL8017973 0.80 CHRM2 (0.41) ALDH1A1KDM4EADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100376564-C Substituted heterocyclic benzoeycloalkenes and the use thereof as substances having analgesic effect GRUENENTHAL CHEMIE (DE) 2008-03-26 CN disclosed
EP-0922703-B1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds GRUENENTHAL GMBH (DE) 2002-12-04 EP disclosed
EP-0922703-A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds Grünenthal GmbH (DE) 1999-06-16 EP disclosed