SCHEMBL7606468

SCHEMBL7606468

CCc1ccc(N2CCN(c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.57
DRD4 P21917 1/20 0.56
KDM4E B2RXH2 4/20 0.56
GAA P10253 2/20 0.56
CHIA Q9BZP6 1/20 0.53
KMT2A Q03164 3/20 0.53
SIGMAR1 Q99720 3/20 0.52
HTR3E A5X5Y0 1/20 0.52
HTR3B O95264 1/20 0.52
ADRB1 P08588 1/20 0.52
HTR3A P46098 1/20 0.52
HTR3D Q70Z44 1/20 0.52
HTR3C Q8WXA8 1/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
ALDH1A1 P00352 1/20 0.50
THRB P10828 1/20 0.50
ME2 P23368 1/20 0.50
ME1 P48163 1/20 0.50
ME3 Q16798 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14438080 0.91 MAPT (0.71) MAPTDRD4KDM4EGAAKMT2A
SCHEMBL28758087 0.89 KDM4E (0.61) MAPTKDM4EGAAKMT2ANPC1
SCHEMBL870704 0.82 HTR3E (0.70) MAPTDRD4KDM4EGAACHIA
SCHEMBL29998630 0.82 HTR3E (0.70) MAPTDRD4KDM4EGAACHIA
SCHEMBL23655782 0.82 ADRB1 (0.53) MAPTKDM4EGAAKMT2AADRB1
SCHEMBL178275 0.82 ALDH1A1 (0.63) MAPTKDM4EGAAKMT2AHTR3A
SCHEMBL12128002 0.82 KDM4E (0.63) MAPTDRD4KDM4ESIGMAR1NPC1
SCHEMBL11164683 0.81 SIGMAR1 (0.51) MAPTDRD4KDM4EGAAKMT2A
SCHEMBL24715763 0.81 KDM4E (0.57) MAPTKDM4EGAAKMT2ANPC1
SCHEMBL2056142 0.81 KDM4E (0.57) MAPTKDM4EGAAKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210340-A1 SUBSTITUTED PIPERAZINE DERIVATIVES, THE PRODUCTION THEREOF AND THEIR UTILIZATION AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 2002-06-05 EP disclosed
WO-2001014355-A1 SUBSTITUTED PIPERAZINE DERIVATIVES, THE PRODUCTION THEREOF AND THEIR UTILIZATION AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-03-01 WO disclosed