SCHEMBL7606900

SCHEMBL7606900

CC(C)OC(=O)Oc1ccc(C(CN(Cc2ccccc2)C(CO)c2ccc(OCc3ccccc3)c(NS(C)(=O)=O)c2)c2ccc(OC(=O)OC(C)C)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 2/20 0.38
TRPV1 Q8NER1 4/20 0.37
CYP19A1 P11511 2/20 0.36
AR P10275 2/20 0.35
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NR3C1 P04150 4/20 0.35
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
ALOX5 P09917 1/20 0.34
ESRRA P11474 1/20 0.34
PTGDR Q13258 1/20 0.34
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606877 0.85 ADRB3 (0.44) ADRB3TRPV1ARNR3C1PGR
SCHEMBL7608285 0.84 ADRB3 (0.40) ADRB3CYP19A1ARNPC1HPGD
SCHEMBL7609423 0.84 ADRB3 (0.40) ADRB3CYP19A1ARNPC1HPGD
SCHEMBL7605292 0.83 ACP1 (0.42) ADRB3TRPV1CYP19A1NR3C1PDE4A
SCHEMBL7604970 0.82 NR3C1 (0.43) ADRB3CYP19A1ARSMN1; SMN2NR3C1
SCHEMBL7610067 0.80 AR (0.38) ADRB3CYP19A1ARNR3C1BRD4
SCHEMBL7611191 0.77 ALDH1A1 (0.44) NPC1RAB9ASMN1; SMN2BRD4
SCHEMBL7605972 0.77 ALDH1A1 (0.44) NPC1HPGDRAB9ASMN1; SMN2ALOX5
SCHEMBL7614703 0.76 SMN1; SMN2 (0.41) CYP19A1ARNPC1RAB9ASMN1; SMN2
SCHEMBL7606168 0.74 PTPN2 (0.41) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed