SCHEMBL7608531

SCHEMBL7608531

COC(=O)Nc1cccc(C(O)(CNCC(O)COc2ccccc2)c2cccc(N(Cc3ccccc3)C(=O)OC)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 14/20 0.42
ADRB3 P13945 12/20 0.42
ADRB2 P07550 7/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7028696 0.79 ADRB1 (0.50) ADRB1ADRB3ADRB2MEN1KMT2A
SCHEMBL7032501 0.76 ALDH1A1 (0.51) ADRB1ADRB3ALDH1A1
SCHEMBL7768357 0.76 ADRB1 (0.44) ADRB1ADRB3ADRB2MEN1KMT2A
SCHEMBL7597017 0.75 MEN1 (0.53) ADRB1ADRB3ADRB2MEN1KMT2A
SCHEMBL7024944 0.75 ADRB1 (0.50) ADRB1ADRB3ADRB2MEN1KMT2A
SCHEMBL7536025 0.71 NPC1 (0.51) ADRB1ADRB3ADRB2MEN1KMT2A
Hydrochloric Acid SCHEMBL7605228 0.70 CYP2D6 (0.55) ADRB1ADRB3ADRB2MEN1KMT2A
SCHEMBL7027312 0.69 MEN1 (0.65) ADRB1ADRB3ADRB2MEN1KMT2A
SCHEMBL7608535 0.68 TSHR (0.41) MEN1KMT2AALDH1A1
SCHEMBL7032860 0.68 SMN1; SMN2 (0.43) MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed