SCHEMBL7609934

SCHEMBL7609934

COc1ccc(C(CCNC(Oc2ccc(O)c(CNS(C)(=O)=O)c2)C(C)O)c2ccc(OC)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 18/20 0.43
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
ADRB2 P07550 3/20 0.39
ADRB1 P08588 2/20 0.39
MITF O75030 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610581 0.85 ADRB2 (0.45) ADRB3CNR1CNR2ADRB2ADRB1
SCHEMBL7609836 0.80 ADRB3 (0.47) ADRB3CNR1CNR2ADRB2ADRB1
SCHEMBL7607623 0.79 ADRB3 (0.44) ADRB3CNR1CNR2ADRB2ADRB1
SCHEMBL7609925 0.79 ADRB3 (0.56) ADRB3ADRB2ADRB1KMT2A
SCHEMBL7607779 0.78 ADRB2 (0.56) ADRB3CNR1CNR2ADRB2ADRB1
SCHEMBL7605258 0.78 ADRB3 (0.47) ADRB3MITFALDH1A1LMNAMAPT
SCHEMBL7608796 0.77 ADRB3 (0.60) ADRB3ADRB2ADRB1
SCHEMBL7610781 0.76 ADRB2 (0.40) ADRB3ADRB2ADRB1
SCHEMBL7610449 0.73 GAA (0.42) ADRB3ADRB2ADRB1MITFALDH1A1
SCHEMBL7606228 0.71 ADRB2 (0.48) ADRB3CNR1CNR2ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed