SCHEMBL7611069

SCHEMBL7611069

COc1ccc(C(CN(Cc2ccccc2)C(CO)c2ccc(OCc3ccccc3)c(N)c2)c2ccc(OC)c(C)c2)cc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
BLM P54132 1/20 0.35
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
F7 P08709 1/20 0.35
F3 P13726 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7611109 0.89 AOC3 (0.40) ALDH1A1NPC1RAB9APOLB
SCHEMBL7610365 0.89 AOC3 (0.40) ALDH1A1NPC1RAB9APOLB
SCHEMBL7606237 0.85 NPC1 (0.39) ALDH1A1NPC1HPGDRAB9ASMN1; SMN2
SCHEMBL7608227 0.85 PTGS1 (0.40) SLC6A2SLC6A3CYP1A2RAB9ASMN1; SMN2
SCHEMBL7606895 0.85 ABCB1 (0.44) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7604970 0.83 NR3C1 (0.43) MEN1KMT2AALDH1A1F2F10
SCHEMBL4728796 0.83 AOC3 (0.39) MEN1KMT2AALDH1A1TRPM8NPC1
SCHEMBL7611061 0.82 MEN1 (0.41) MEN1KMT2AALDH1A1TRPM8SLC6A2
SCHEMBL7606221 0.82 NPC1 (0.46) MEN1KMT2ATRPM8KDM4EF2
SCHEMBL7611531 0.80 ESR1 (0.38) ALDH1A1TRPM8KDM4ENPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed