SCHEMBL7616686

SCHEMBL7616686

COc1ccc(P(=O)(c2ccccc2)c2ccccc2)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.51
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP1A1 P04798 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP1B1 Q16678 1/20 0.44
LMNA P02545 1/20 0.44
MEN1 O00255 3/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
NQO2 P16083 1/20 0.43
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
CA12 O43570 3/20 0.43
CA9 Q16790 3/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA7 P43166 2/20 0.43
CA14 Q9ULX7 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7712023 0.84 GRM4 (0.46) KMT2AHTTL3MBTL1LMNAMEN1
SCHEMBL7622693 0.81 TUBB4A (0.49) KMT2AHTTL3MBTL1CYP1A2MEN1
SCHEMBL28453272 0.78 L3MBTL1 (0.44) KMT2AHTTL3MBTL1CYP1A1CYP1A2
SCHEMBL14754995 0.77 KMT2A (0.62) KMT2AHTTL3MBTL1LMNAMEN1
SCHEMBL5619254 0.76 CA4 (0.54) KMT2AHTTLMNAMEN1NPC1
SCHEMBL5619896 0.76 CA4 (0.54) KMT2AHTTLMNAMEN1NPC1
SCHEMBL7619840 0.76 LMNA (0.50) KMT2AHTTL3MBTL1LMNAMEN1
SCHEMBL11225829 0.75 CA2 (0.45) KMT2AHTTL3MBTL1CYP1A2LMNA
SCHEMBL10723400 0.75 CA2 (0.45) KMT2AHTTL3MBTL1CYP1A2LMNA
SCHEMBL4406229 0.75 TSHR (0.48) KMT2AL3MBTL1CYP1A2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0926152-B1 Process for the manufacture of bis(phosphine oxide)-and bis(phosphonate)-compounds HOFFMANN LA ROCHE (CH) 2002-09-11 EP disclosed
US-6162929-A Process for the manufacture of bisphosphine oxide and bisphosphonate compounds HOFFMANN-LA ROCHE INC. (US) 2000-12-19 US disclosed
EP-0926152-A1 Process for the manufacture of bis(phosphine oxide)-and bis(phosphonate)-compounds F. HOFFMANN-LA ROCHE AG (CH) 1999-06-30 EP disclosed
US-5488172-A Chiral phosphorus compounds HOFFMANN-LA ROCHE INC. (US) 1996-01-30 US disclosed
EP-0398132-B1 Phosphorous compounds HOFFMANN LA ROCHE (CH) 1995-09-20 EP disclosed
EP-0398132-A2 Phosphorous compounds F. HOFFMANN-LA ROCHE AG (CH) 1990-11-22 EP disclosed