SCHEMBL762541

SCHEMBL762541

CCCCn1c([C@@H]2CCCN(C(=O)C[C@H](C)Cc3ccc4ccccc4c3)C2)nc2cccc(C)c21

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 7/20 0.38
CYP2D6 P10635 6/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
KCNH2 Q12809 7/20 0.36
PROKR1 Q8TCW9 1/20 0.36
CHRM1 P11229 2/20 0.35
TLR8 Q9NR97 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763431 0.92 HRH1 (0.38) HRH1CYP2D6NPC1RAB9AKCNH2
SCHEMBL762543 0.88 CYP2D6 (0.36) HRH1CYP2D6NPC1RAB9AKCNH2
SCHEMBL762535 0.86 HRH1 (0.40) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL740700 0.84 KCNH2 (0.36) HRH1CYP2D6NPC1RAB9AKCNH2
SCHEMBL740699 0.84 KCNH2 (0.36) HRH1CYP2D6NPC1RAB9AKCNH2
SCHEMBL762548 0.84 KCNH2 (0.40) HRH1CYP2D6NPC1RAB9AKCNH2
SCHEMBL762546 0.80 KCNH2 (0.37) HRH1CYP2D6KCNH2CHRM1
SCHEMBL762831 0.80 TLR8 (0.36) HRH1CYP2D6NPC1RAB9AKCNH2
SCHEMBL742487 0.79 HRH1 (0.36) HRH1CYP2D6KCNH2PROKR1CHRM1
SCHEMBL763816 0.79 CTSB (0.36) HRH1CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed