SCHEMBL7646276

SCHEMBL7646276

O=[N+]([O-])c1[c]ccc(C(F)(F)F)c1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCC8 Q09428 4/20 0.36
KCNJ11 Q14654 4/20 0.36
EPAS1 Q99814 2/20 0.33
VEGFA P15692 1/20 0.33
KIF11 P52732 1/20 0.32
AR P10275 7/20 0.31
ALDH1A1 P00352 2/20 0.31
SIRT6 Q8N6T7 1/20 0.31
PDE7A Q13946 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27913942 0.81 ABCC8 (0.33) ABCC8KCNJ11EPAS1VEGFAKIF11
SCHEMBL3556690 0.76 ALDH1A1 (0.34) EPAS1KIF11ARALDH1A1SIRT6
SCHEMBL301080 0.76 TDP1 (0.34) ALDH1A1TDP1
SCHEMBL18478 0.73 TSHR (0.42) ALDH1A1TDP1
SCHEMBL1995800 0.72 TDP1 (0.46) ABCC8KCNJ11EPAS1VEGFAKIF11
SCHEMBL9789548 0.72 ALDH1A1 (0.42) ALDH1A1TDP1
SCHEMBL3047388 0.72 GPR35 (0.46) ALDH1A1TDP1
SCHEMBL6514635 0.71 AR (0.38) KIF11ARALDH1A1SIRT6TDP1
SCHEMBL11690136 0.69 ALDH1A1 (0.33) ALDH1A1TDP1
SCHEMBL10731966 0.69 ALDH1A1 (0.39) ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6486153-B1 Phenylindole derivatives as 5-HT2A receptor ligands MERCK SHARP & DOHME LTD. 2002-11-26 US disclosed
WO-1999011619-A1 PHENYLINDOLE DERIVATIVES AS 5-HT2A RECEPTOR LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1999-03-11 WO disclosed