SCHEMBL7649652

SCHEMBL7649652

CN1Cc2cc([N+](=O)[O-])ccc2CC1(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
TSHR P16473 2/20 0.43
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TDP2 O95551 1/20 0.43
DPP7 Q9UHL4 1/20 0.42
PNMT P11086 5/20 0.42
ADRA2A P08913 3/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 3/20 0.42
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
TLR9 Q9NR96 1/20 0.42
SIRT6 Q8N6T7 1/20 0.41
HTT P42858 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1952644 0.79 TDP2 (0.44) LMNATSHRALDH1A1TDP1TDP2
SCHEMBL29945643 0.78 DPP7 (0.50) LMNATSHRALDH1A1TDP1TDP2
SCHEMBL7657931 0.76 DPP7 (0.41) LMNATDP2DPP7PNMTADRA2A
SCHEMBL29558059 0.74 ADRA2A (0.51) LMNAALDH1A1PNMTADRA2AL3MBTL1
SCHEMBL324724 0.74 ADRA2A (0.51) LMNAALDH1A1PNMTADRA2AL3MBTL1
SCHEMBL7656239 0.73 NR1H2 (0.35) LMNAALDH1A1ADRA2CMAPTMEN1
SCHEMBL5917126 0.73 CA1 (0.47) LMNATSHRALDH1A1TDP1TDP2
Hydrochloric Acid SCHEMBL7832321 0.73 ADRA2A (0.50) LMNAALDH1A1PNMTADRA2AL3MBTL1
SCHEMBL8607529 0.73 MAPT (0.46) LMNAALDH1A1TDP1DPP7MAPT
SCHEMBL25339488 0.73 SIRT6 (0.44) LMNAALDH1A1TDP1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed
EP-1104404-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2001-06-06 EP disclosed
WO-2000009486-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSIVANTS SMITHKLINE BEECHAM P.L.C. (GB) 2000-02-24 WO disclosed