SCHEMBL7650106

SCHEMBL7650106

CNC(=O)[C@@H](Cc1ccccc1)NC[C@@H](Cc1ccc2ccccc2c1)NC(=O)O

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FCER2 P06734 5/20 0.59
MMP9 P14780 5/20 0.50
MMP8 P22894 5/20 0.50
MMP2 P08253 2/20 0.50
MME P08473 2/20 0.48
ACE P12821 2/20 0.48
CPA1 P15085 2/20 0.48
ACE2 Q9BYF1 2/20 0.48
TACR1 P25103 1/20 0.47
CTSB P07858 3/20 0.46
CTSS P25774 3/20 0.46
CTSL P07711 2/20 0.46
CTSK P43235 2/20 0.44
PLAT P00750 1/20 0.43
PSMB1 P20618 1/20 0.43
PSMB5 P28074 1/20 0.43
PSMB2 P49721 1/20 0.43
MMP1 P03956 1/20 0.43
OPRD1 P41143 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651306 1.00 FCER2 (0.59) FCER2MMP9MMP8MMP2MME
SCHEMBL7646980 0.87 CTSS (0.60) FCER2MMP9MMP8MMP2ACE
SCHEMBL7646982 0.87 CTSS (0.60) FCER2MMP9MMP8MMP2ACE
SCHEMBL29203892 0.78 MME (0.51) FCER2MMEACECPA1ACE2
SCHEMBL8206981 0.78 FCER2 (0.60) FCER2MMP9MMP8MMP2MME
SCHEMBL7650909 0.75 FCER2 (0.46) FCER2MMP9MMP8MMP2MME
SCHEMBL21988101 0.75 MMP1 (0.63) FCER2MMP9MMP8MMP2MMP1
SCHEMBL6851903 0.74 FCER2 (1.00) FCER2MMP9MMP8MMP2MMP1
SCHEMBL6434826 0.74 MMP2 (0.73) FCER2MMP9MMP8MMP2MME
SCHEMBL7965979 0.73 FCER2 (0.61) FCER2MMP9MMP8MMP2MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1184370-A2 Compounds with growth hormone releasing properties NOVO NORDISK A/S (DK) 2002-03-06 EP disclosed
US-6274584-B1 PEPTIDE DERIVATIVES; BIOAVAILABILITY; ENZYME RESISTANCE; MILK AND WOOL PRODUCTION NOVO NORDISK A/S (DK) 2001-08-14 US disclosed
US-6127354-A FOR TREATMENT OF GROWTH DISORDERS OR TO STIMULATE PRODUCTION OF WOOL OR MILK NOVO NORDISK A/S (DK) 2000-10-03 US disclosed
US-5922770-A NOVEL COMPOUNDS THAT STIMULATE THE RELEASE OF GROWTH HORMONE FROM THE PITUITARY NOVO NORDISK A/S (DK) 1999-07-13 US disclosed
EP-0923539-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1999-06-23 EP disclosed
WO-1998003473-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1998-01-29 WO disclosed