SCHEMBL7650322

SCHEMBL7650322

CC(C)(C(=O)OCC(=O)c1ccccc1)n1c(=O)[nH]c2cc(F)c(F)cc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 2/20 0.38
USP2 O75604 1/20 0.37
KDM4E B2RXH2 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
HPGD P15428 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
TSHR P16473 1/20 0.34
CTSV O60911 1/20 0.34
CTSL P07711 1/20 0.34
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7650012 0.89 MPO (0.44) SMN1; SMN2POLBMAPTKDM4EL3MBTL1
SCHEMBL7648323 0.88 SMN1; SMN2 (0.41) SMN1; SMN2POLBMAPTKDM4EL3MBTL1
SCHEMBL7655615 0.86 SMN1; SMN2 (0.45) SMN1; SMN2POLBMAPTUSP2KDM4E
SCHEMBL7652031 0.84 CA12 (0.44) SMN1; SMN2POLBMAPTKDM4EL3MBTL1
SCHEMBL7649499 0.84 CA9 (0.45) SMN1; SMN2POLBMAPTUSP2KDM4E
SCHEMBL7648338 0.83 FEN1 (0.45) SMN1; SMN2POLBMAPTUSP2KDM4E
SCHEMBL7651849 0.82 MPO (0.38) SMN1; SMN2POLBMAPTKDM4EALDH1A1
SCHEMBL7653637 0.77 MPO (0.43) POLBKDM4EALDH1A1CA12CA9
SCHEMBL7650555 0.74 ALDH1A1 (0.35) SMN1; SMN2USP2ALDH1A1NPC1RAB9A
SCHEMBL7653151 0.73 KDM4E (0.44) SMN1; SMN2MAPTUSP2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed