SCHEMBL7650467

SCHEMBL7650467

CCOc1cc(O)c[c]c1Oc1ccc(OCCN2CCCCC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.57
PSMB1 P20618 7/20 0.47
PSMB5 P28074 7/20 0.47
PSMB2 P49721 4/20 0.47
ALDH1A1 P00352 1/20 0.47
LTA4H P09960 6/20 0.47
PTGS2 P35354 3/20 0.46
PTGS1 P23219 1/20 0.46
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7108553 0.90 KDM4E (0.49) KDM4EPSMB1PSMB5PSMB2LTA4H
SCHEMBL3130426 0.85 LTA4H (0.52) PSMB1PSMB5PSMB2LTA4HPTGS2
SCHEMBL7777295 0.84 LTA4H (0.53) PSMB1PSMB5PSMB2LTA4HPTGS2
SCHEMBL7778580 0.79 LTA4H (0.53) PSMB1PSMB5PSMB2LTA4HPTGS2
SCHEMBL7505643 0.78 SMN1; SMN2 (0.47) KDM4EALDH1A1LTA4HESR1ESR2
SCHEMBL7918786 0.76 LTA4H (0.47) KDM4EPSMB1PSMB5PSMB2LTA4H
SCHEMBL13297167 0.75 KDM4E (0.82) KDM4EPSMB1PSMB5PSMB2ALDH1A1
SCHEMBL7441879 0.75 TDP1 (0.52) KDM4EALDH1A1ESR1ESR2
SCHEMBL7212312 0.74 PSMB1 (0.49) KDM4EPSMB1PSMB5PSMB2ALDH1A1
SCHEMBL7466056 0.74 LTA4H (0.61) KDM4EALDH1A1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204656-A2 A CRYSTALLINE FORM OF 6-HYDROXY-3-(4-[2-(PIPERIDIN-1-YL) ETHOXY] PHENOXY)-2-(4-METHOXYPHENYL) BENZO[B]THIOPHENE HYDROCHLORIDE ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2001009116-A2 A NOVEL CRYSTALLINE FORM OF 6-HYDROXY-3- (4-[2-(PIPERIDIN-1-YL) ETHOXY]PHENOXY)- 2-(4-METHOXYPHENYL)BENZO[b]THIOPHENE HYDROCHLORIDE ELI LILLY AND COMPANY (US) 2001-02-08 WO disclosed