SCHEMBL7651049

SCHEMBL7651049

CCOC(=O)C(C)(C)n1c(=O)[nH]c2cccc(F)c2c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.51
GAA P10253 2/20 0.38
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DAO P14920 1/20 0.38
ADORA3 P0DMS8 2/20 0.37
NLRP3 Q96P20 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
HSD17B10 Q99714 2/20 0.36
GLA P06280 1/20 0.36
HPGD P15428 1/20 0.36
MAP3K5 Q99683 1/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7648338 0.85 FEN1 (0.45) FEN1NPC1SMN1; SMN2DAOKDM4E
SCHEMBL7650006 0.82 FEN1 (0.58) FEN1DAO
SCHEMBL7652236 0.80 SMN1; SMN2 (0.55) FEN1GAANPC1SMN1; SMN2ADORA3
SCHEMBL7651849 0.78 MPO (0.38) GAANPC1SMN1; SMN2DAOADORA3
SCHEMBL7651932 0.76 FEN1 (0.51) FEN1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL7653151 0.74 KDM4E (0.44) GAANPC1SMN1; SMN2ADORA3KDM4E
SCHEMBL30970862 0.74 FEN1 (0.60) FEN1SMN1; SMN2DAOADORA3KDM4E
SCHEMBL7653163 0.73 SMN1; SMN2 (0.54) NPC1SMN1; SMN2KDM4EALDH1A1TSHR
SCHEMBL7649595 0.73 KDM4E (0.47) GAANPC1SMN1; SMN2KDM4EALDH1A1
SCHEMBL10507746 0.72 FEN1 (0.66) FEN1DAOADORA3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed