SCHEMBL7651581

SCHEMBL7651581

COc1ccc(CSCCCC(=N)C(=O)N(N)C=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
PKM P14618 1/20 0.44
IDO1 P14902 2/20 0.41
MAPT P10636 2/20 0.38
ALOX5 P09917 1/20 0.38
ATM Q13315 1/20 0.38
GAA P10253 1/20 0.37
SAE1 Q9UBE0 1/20 0.36
UBA2 Q9UBT2 1/20 0.36
GLA P06280 1/20 0.36
DAO P14920 1/20 0.36
EPHX1 P07099 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7647968 0.76 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2PKMIDO1MAPT
SCHEMBL16334693 0.71 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2PKMMAPTALOX5
SCHEMBL17045908 0.71 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2PKMMAPTGAA
SCHEMBL7355822 0.70 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2PKMIDO1MAPT
SCHEMBL8003157 0.70 CYP2C19 (0.64) ALDH1A1SMN1; SMN2PKMIDO1GAA
SCHEMBL530979 0.70 PDE4B (0.54) ALDH1A1SMN1; SMN2PKMGAAEPHX1
SCHEMBL7604958 0.69 EPHX1 (0.43) ALDH1A1SMN1; SMN2IDO1ALOX5GAA
SCHEMBL17045933 0.69 HDAC1 (0.59) ALDH1A1SMN1; SMN2PKM
SCHEMBL7651583 0.68 ALOX5 (0.41) ALDH1A1SMN1; SMN2PKMIDO1ALOX5
SCHEMBL9043314 0.68 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2PKMIDO1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212096-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME Brenner, Sydney (US) 2002-06-12 EP disclosed
WO-2001013958-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME BRENNER SYDNEY (US) 2001-03-01 WO disclosed