SCHEMBL7651583

SCHEMBL7651583

COc1ccc(CSN=CCCCC(=O)N(N)C=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.41
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
IDO1 P14902 2/20 0.36
ALDH1A1 P00352 4/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
EPHX1 P07099 1/20 0.35
CNR1 P21554 2/20 0.34
KDM4E B2RXH2 1/20 0.34
CNR2 P34972 1/20 0.34
F2RL1 P55085 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HTT P42858 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
PKM P14618 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7604958 0.76 EPHX1 (0.43) ALOX5BCHEACHEIDO1ALDH1A1
SCHEMBL7651581 0.68 ALDH1A1 (0.44) ALOX5IDO1ALDH1A1EPHX1SMN1; SMN2
SCHEMBL6122244 0.61 TSHR (0.65) ALOX5BCHEACHEALDH1A1F2RL1
SCHEMBL6121660 0.61 TSHR (0.65) ALOX5BCHEACHEALDH1A1F2RL1
SCHEMBL31329297 0.60 ALOX5 (0.82) ALOX5BCHEACHEALDH1A1CYP3A4
SCHEMBL6122069 0.60 TSHR (0.63) ALOX5BCHEACHEALDH1A1F2RL1
SCHEMBL10691859 0.60 ALOX5 (1.00) ALOX5BCHEACHEALDH1A1F2RL1
SCHEMBL6121985 0.60 TSHR (0.63) ALOX5BCHEACHEALDH1A1F2RL1
SCHEMBL9973241 0.60 IDO1 (0.44) ALOX5IDO1ALDH1A1EPHX1F2RL1
SCHEMBL10823756 0.59 IDO1 (0.59) ALOX5IDO1ALDH1A1EPHX1F2RL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212096-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME Brenner, Sydney (US) 2002-06-12 EP disclosed
WO-2001013958-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME BRENNER SYDNEY (US) 2001-03-01 WO disclosed