SCHEMBL7604958

SCHEMBL7604958

COc1ccc(CSC(N)CCCC(=O)N(N)C=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.43
ALOX5 P09917 2/20 0.42
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
IDO1 P14902 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.37
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
POLB P06746 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LDHA P00338 1/20 0.35
F2RL1 P55085 1/20 0.35
HTT P42858 1/20 0.34
ANPEP P15144 1/20 0.34
ERAP2 Q6P179 1/20 0.34
LTB4R Q15722 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7604900 0.80 EPHX1 (0.45) EPHX1ALOX5IDO1L3MBTL1GAA
SCHEMBL7651583 0.76 ALOX5 (0.41) EPHX1ALOX5BCHEACHEIDO1
SCHEMBL8932479 0.72 TAAR1 (0.50) EPHX1BCHEACHEIDO1ALDH1A1
SCHEMBL7651581 0.69 ALDH1A1 (0.44) EPHX1ALOX5IDO1GAAALDH1A1
SCHEMBL7088679 0.65 SLC6A4 (0.58) EPHX1BCHEACHEIDO1L3MBTL1
SCHEMBL6121660 0.64 TSHR (0.65) ALOX5BCHEACHEL3MBTL1ALDH1A1
SCHEMBL5971492 0.64 SLC6A4 (0.53) EPHX1BCHEACHEIDO1ALDH1A1
SCHEMBL7881281 0.64 SLC6A4 (0.52) EPHX1BCHEACHEIDO1ALDH1A1
SCHEMBL6122069 0.63 TSHR (0.63) ALOX5BCHEACHEL3MBTL1ALDH1A1
SCHEMBL7346371 0.63 L3MBTL1 (0.62) EPHX1IDO1L3MBTL1GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212096-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME Brenner, Sydney (US) 2002-06-12 EP disclosed
WO-2001013958-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME BRENNER SYDNEY (US) 2001-03-01 WO disclosed