SCHEMBL7653872

SCHEMBL7653872

CC(C)c1ccc(C(=O)Nc2ccc3c(c2)CNC(C)(C)C3)cc1C#N

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
PKN2 Q16513 1/20 0.38
MELK Q14680 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
EZH2 Q15910 1/20 0.36
MCHR1 Q99705 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656532 0.82 ROCK2 (0.43) ROCK2
SCHEMBL7993332 0.78 ROCK2 (0.45) ROCK2CYP3A4CYP2C19ALDH1A1
SCHEMBL7656595 0.77 ROCK2 (0.39) ROCK2
SCHEMBL6295077 0.77 ROCK2 (0.58) ROCK2CYP3A4
Hydrochloric Acid SCHEMBL6299497 0.76 ROCK2 (0.57) ROCK2CYP3A4
SCHEMBL7659472 0.76 ROCK2 (0.43) ROCK2CYP3A4NPC1ALDH1A1MAPT
SCHEMBL7659693 0.75 MEN1 (0.44) CYP3A4CYP2C19NPC1ALDH1A1MAPT
SCHEMBL7658184 0.75 RORC (0.49) ROCK2NPC1ALDH1A1MAPTRAB9A
SCHEMBL7656812 0.75 CYP26A1 (0.38) ROCK2CYP3A4CYP2C19NPC1ALDH1A1
SCHEMBL7658566 0.72 MAPT (0.58) CYP3A4CYP2C19NPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US claimed
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed