SCHEMBL7656595

SCHEMBL7656595

CC(C)c1ccc(C(=O)Nc2ccc3c(c2)CN(C(=O)C(F)(F)F)C(C)(C)C3)cc1C#N

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.39
NAMPT P43490 7/20 0.39
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
KCNE1 P15382 1/20 0.36
KCNQ1 P51787 1/20 0.36
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656532 0.86 ROCK2 (0.43) ROCK2NAMPT
SCHEMBL7650167 0.79 ROCK2 (0.45) ROCK2KCNQ3KCNQ2
SCHEMBL7649708 0.78 KMT2A (0.41) ROCK2KCNQ3KCNQ2
SCHEMBL6295077 0.78 ROCK2 (0.58) ROCK2
SCHEMBL7653872 0.77 ROCK2 (0.38) ROCK2
Hydrochloric Acid SCHEMBL6299497 0.77 ROCK2 (0.57) ROCK2
SCHEMBL7993332 0.77 ROCK2 (0.45) ROCK2NAMPT
SCHEMBL7655163 0.76 MAPT (0.46) ROCK2NAMPT
SCHEMBL7652124 0.76 MAPT (0.52)
SCHEMBL7659472 0.73 ROCK2 (0.43) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US claimed
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed