SCHEMBL7654909

SCHEMBL7654909

Cc1ccc2c(c1)c(=O)n(C(C)(C)C(=O)OCC(=O)c1ccccc1)c(=O)n2CCCCBr

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
PGR P06401 1/20 0.39
RORA P35398 1/20 0.39
RORC P51449 1/20 0.39
RORB Q92753 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
CNR2 P34972 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
KMT2A Q03164 1/20 0.34
TNF P01375 1/20 0.34
PNP P00491 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7650485 0.90 HDAC1 (0.38) SMN1; SMN2PTGDR2ALDH1A1L3MBTL1CNR2
SCHEMBL7651760 0.90 PTGDR2 (0.40) PTGDR2CNR2KMT2A
SCHEMBL7651131 0.90 CNR2 (0.42) SMN1; SMN2ALDH1A1L3MBTL1CNR2KDM4E
SCHEMBL7653503 0.88 ALDH1A1 (0.37) POLBSMN1; SMN2ALDH1A1CNR2HTT
SCHEMBL7651232 0.88 RORA (0.41) POLBSMN1; SMN2PGRRORARORC
SCHEMBL7650555 0.87 ALDH1A1 (0.35) SMN1; SMN2NPC1RAB9AALDH1A1CNR2
SCHEMBL7649498 0.85 HDAC6 (0.40) SMN1; SMN2ALDH1A1L3MBTL1CNR2KDM4E
SCHEMBL7651764 0.80 ALDH1A1 (0.35) SMN1; SMN2NPC1RAB9AALDH1A1CNR2
SCHEMBL7655134 0.80 TNF (0.51) NPC1ALDH1A1L3MBTL1CNR2KDM4E
SCHEMBL7651781 0.79 KCNA3 (0.39) POLBSMN1; SMN2ALDH1A1L3MBTL1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed