SCHEMBL7655147

SCHEMBL7655147

CCOC(=O)CCn1c(CC(=O)OCC)nc2c(N3CCCCC3)cccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.45
NPY1R P25929 2/20 0.40
HPGD P15428 1/20 0.40
TP53 P04637 1/20 0.40
LMNA P02545 2/20 0.37
ALDH1A1 P00352 2/20 0.37
TSHR P16473 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
AKT1 P31749 1/20 0.37
CTNNB1 P35222 1/20 0.37
MAPT P10636 2/20 0.37
PKM P14618 1/20 0.37
NOTUM Q6P988 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CXCR3 P49682 1/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
CREBBP Q92793 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778204 0.90 HTR6 (0.42) CNR2NPY1RIRAK4
SCHEMBL5774251 0.88 ALDH1A1 (0.41) CNR2NPY1RHPGDTP53LMNA
SCHEMBL5776881 0.86 ALDH1A1 (0.43) CNR2NPY1RALDH1A1MAPTTMEM97
SCHEMBL5775304 0.80 ALDH1A1 (0.43) NPY1RHPGDLMNAALDH1A1TSHR
SCHEMBL5775785 0.76 KCNH2 (0.41) CNR2NPY1RALDH1A1MAPT
SCHEMBL7419269 0.74 NPY1R (0.35) CNR2NPY1RCTNNB1IRAK4
SCHEMBL5777998 0.70 ALDH1A1 (0.43) HPGDTP53LMNAALDH1A1TSHR
SCHEMBL4887137 0.67 HTR1A (0.38) ALDH1A1MAPTTMEM97SIGMAR1
SCHEMBL7806454 0.67 MAPT (0.41) CNR2NPY1RHPGDLMNAALDH1A1
SCHEMBL7978871 0.67 AKT1 (0.42) HPGDALDH1A1TSHRAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358946-B1 ANTIDEPRESSANTS, ANXIOLYTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS, ANTICONVULSANTS, AND HYPNOSIS AGENTS; SLEEP DISORDER TREATMENT ORTHO-MCNEIL PHARMACEUTICAL, INC. 2002-03-19 US disclosed