SCHEMBL7419269

SCHEMBL7419269

CCOC(=O)CCn1c(CC(=O)OCC)nc2c(N3CCNCC3C(=O)OCCCCF)cccc21

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 2/20 0.35
CNR2 P34972 2/20 0.33
CTNNB1 P35222 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414507 0.92 NPY1R (0.32) NPY1R
SCHEMBL5778204 0.78 HTR6 (0.42) NPY1RCNR2IRAK4
SCHEMBL7655147 0.74 CNR2 (0.45) NPY1RCNR2CTNNB1IRAK4
SCHEMBL5776881 0.68 ALDH1A1 (0.43) NPY1RCNR2
SCHEMBL7429443 0.65 MEN1 (0.45)
SCHEMBL5774251 0.65 ALDH1A1 (0.41) NPY1RCNR2
SCHEMBL8944811 0.63 MAPT (0.49)
SCHEMBL16927639 0.62 CHEK1 (0.55)
SCHEMBL5401386 0.62 TACR1 (0.48)
SCHEMBL5408982 0.62 TACR1 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1200433-A1 C-6 RING-SUBSTITUTED PYRIDO 1,2- i a /i ]BENZIMIDAZOLE DERIVATIVES USEFUL IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS Ortho-McNeil Pharmaceutical, Inc. (US) 2002-05-02 EP disclosed
WO-2001009132-A1 C-6 RING-SUBSTITUTED PYRIDO[1,2-a]BENZIMIDAZOLE DERIVATIVES USEFUL IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-02-08 WO disclosed