SCHEMBL7657325

SCHEMBL7657325

Cc1ccc(-n2nc(-c3ccccc3)n(C)c2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.54
MAPT P10636 2/20 0.52
POLB P06746 2/20 0.48
THRB P10828 1/20 0.45
ADORA2A P29274 2/20 0.44
ADORA2B P29275 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HIF1A Q16665 1/20 0.43
TP53 P04637 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7658278 0.94 MAPT (0.52) ADORA3MAPTPOLBTHRBALDH1A1
SCHEMBL7652545 0.92 ADORA3 (0.49) ADORA3MAPTADORA2AADORA2BALDH1A1
SCHEMBL7652943 0.83 RPA1 (0.52) ADORA3MAPTADORA2AALDH1A1TP53
SCHEMBL5820957 0.81 TP53 (0.46) ADORA3MAPTPOLBALDH1A1TP53
SCHEMBL7682175 0.79 ALDH1A1 (0.55) ADORA3MAPTALDH1A1
SCHEMBL7655309 0.79 CA1 (0.45) ADORA3MAPTPOLBALDH1A1TP53
SCHEMBL7649140 0.79 TP53 (0.58) ADORA3MAPTPOLBADORA2AALDH1A1
SCHEMBL7650590 0.79 KDM4E (0.49) MAPTPOLBADORA2AALDH1A1ADORA1
SCHEMBL7650966 0.78 ADORA3 (0.45) ADORA3MAPTADORA2AALDH1A1ADORA1
SCHEMBL7659194 0.77 ALDH1A1 (0.51) MAPTPOLBADORA2AADORA2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492407-B2 NEUROPROTECTIVE ACTIVITY BOEHRINGER IMGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed