SCHEMBL7657773

SCHEMBL7657773

CC(=O)Cc1cc[nH]c(=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 7/20 0.40
NSD2 O96028 1/20 0.38
ABL1 P00519 1/20 0.38
PPARG P37231 1/20 0.38
RIN1 Q13671 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
NOTUM Q6P988 1/20 0.37
POLB P06746 1/20 0.37
HPGDS O60760 1/20 0.36
GPR84 Q9NQS5 1/20 0.35
VNN1 O95497 1/20 0.34
GRM2 Q14416 1/20 0.34
GRM3 Q14832 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
ALDH1A1 P00352 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18460841 0.81 NSD2 (0.36) ALDH2NSD2ABL1PPARGRIN1
SCHEMBL4604293 0.81 CA2 (0.44) ALDH2NSD2ABL1PPARGRIN1
SCHEMBL21550134 0.80 ALDH1A1 (0.49) ALDH2NSD2ABL1PPARGRIN1
SCHEMBL4161939 0.78 SMN1; SMN2 (0.49) ALDH2L3MBTL1ALDH1A1
SCHEMBL2837445 0.76 NSD2 (0.37) ALDH2NSD2ABL1PPARGRIN1
SCHEMBL1161397 0.75
SCHEMBL885378 0.75
SCHEMBL6929568 0.73
SCHEMBL13660763 0.72 GPR84 (0.43) ALDH2NSD2ABL1PPARGRIN1
SCHEMBL22229971 0.72 KEAP1 (0.48) NSD2ABL1PPARGRIN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436951-B1 3-HYDROXY-3-(4-OXO-4,6-DIHYDROINDOLIZINO (1,2-B) QUINOLINE-2-YL) PENTANOIC ACID, INHIBITING TOPOISOMERASE I AND/OR II; ANTITUMOR, PARASITICIDE; REACTING A PYRIDINONE WITH A QUINOLINE, CYCLIZATION, EPOXIDATION SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2002-08-20 US disclosed
EP-1042323-A1 NOVEL CAMPTOTHECIN TETRACYCLIC ANALOGUES, PREPARATION, METHODS, APPLICATIONS AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2000-10-11 EP disclosed
WO-1999033829-A1 NOVEL CAMPTOTHECIN TETRACYCLIC ANALOGUES, PREPARATION, METHODS, APPLICATIONS AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1999-07-08 WO disclosed