SCHEMBL7665337

SCHEMBL7665337

CSC1=NC(C)(c2ccccc2)C(=O)N1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
DHFR P00374 3/20 0.38
TSHR P16473 1/20 0.35
LMNA P02545 1/20 0.34
ELANE P08246 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HBB P68871 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
MMP2 P08253 1/20 0.33
MMP13 P45452 1/20 0.33
PKM P14618 1/20 0.32
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484402 0.77 ELANE (0.50) ALDH1A1LMNAELANEKDM4EMAPT
SCHEMBL9234331 0.72 SIRT1 (0.46) MAPTMMP2MMP13PKM
SCHEMBL7651737 0.70 ALDH1A1 (0.35) ALDH1A1MAPTBACE1BACE2
Fenamidone SCHEMBL550975 0.69 CYP1A2 (0.38) ALDH1A1LMNAMAPTBACE1BACE2
Fenamidone SCHEMBL15286728 0.69 CYP1A2 (0.38) ALDH1A1LMNAMAPTBACE1BACE2
Fenamidone SCHEMBL17701153 0.68 CYP1A2 (0.37) ALDH1A1LMNAMAPTBACE1BACE2
SCHEMBL7475363 0.68 ALDH1A1 (0.33) ALDH1A1MEN1MAPTKMT2ABACE1
SCHEMBL9231712 0.65 CYP1A2 (0.32) ALDH1A1LMNAELANEKDM4EMEN1
SCHEMBL9234360 0.65 CYP1A2 (0.32) ALDH1A1MEN1MAPTKMT2A
SCHEMBL30942995 0.65 ALDH1A1 (0.59) ALDH1A1DHFRTSHRELANEMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344564-B1 FUNGICIDES RHONE-POULENC, INC. 2002-02-05 US disclosed
US-6018052-A APPLYING TO CROPS OR THEIR SEEDS TO PREVENT OR CURE FUNGAL DISEASES; STEREOSPECIFIC COMPOUND WITH IMPROVED BIOLOGICAL ACTIVITY RHONE-POULENC AGROCHIMIE (FR) 2000-01-25 US disclosed
US-6002016-A Fungicidal 2-imidazolin-5-ones and 2-imidazoline-5-thiones RHONE-POULENC AGROCHIMIE (FR) 1999-12-14 US disclosed
US-5650519-A Optically active 5, 5-disubstituted-3-(mono- or disubstituted amino)-2-thiohydantoin intermediates to fungicidal 2-imidazolin-5-ones RHONE-POULENC AGROCHIMIE (FR) 1997-07-22 US disclosed
US-5637729-A AGRICULTURE RHONE-POULENC AGROCHIMIE (FR) 1997-06-10 US disclosed
EP-0551048-A1 2-imidazoline-5-one and 2-imidazoline-5-thiones derivatives as fungizides RHONE-POULENC AGROCHIMIE (FR) 1993-07-14 EP disclosed