SCHEMBL7668656

SCHEMBL7668656

CCCCC(NC(=O)c1ccc(NC(=O)c2ccc3ccccc3c2)cc1)C(=O)CNC(C)=O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.52
CCKBR P32239 1/20 0.49
CASP1 P29466 3/20 0.48
RAB9A P51151 6/20 0.47
NPC1 O15118 5/20 0.47
CASP3 P42574 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
DEGS1 O15121 1/20 0.47
NR1H4 Q96RI1 1/20 0.46
PLAU P00749 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7659961 0.92 MEN1 (0.52) KMT2AMEN1CCKBRCASP1RAB9A
SCHEMBL7659998 0.90 MEN1 (0.45) KMT2AMEN1CCKBRCASP1RAB9A
SCHEMBL7654043 0.84 ALDH1A1 (0.54) KMT2ACCKBRPLAUHDAC3HDAC1
SCHEMBL7668106 0.83 CASP1 (0.46) KMT2AMEN1CCKBRCASP1RAB9A
SCHEMBL7385051 0.82 PTPN1 (0.46) CCKBRRAB9ANPC1HDAC3HDAC1
SCHEMBL7666410 0.81 CCKBR (0.42) KMT2AMEN1CCKBRCASP1RAB9A
SCHEMBL7658785 0.79 ALDH1A1 (0.45) KMT2AMEN1CCKBRPLAUHDAC3
SCHEMBL7665000 0.77 ALDH1A1 (0.52) KMT2AMEN1CCKBRPLAUHDAC3
SCHEMBL7428036 0.76 CA2 (0.45) CCKBRRAB9ANPC1HDAC3HDAC1
SCHEMBL7664997 0.74 PTPN1 (0.51) KMT2AMEN1CCKBRRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed