SCHEMBL7675073

SCHEMBL7675073

COc1nc2cc(Cl)c(Cl)c(-c3nn[nH]c3-c3ccccc3)c2nc1OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
NFKB1 P19838 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NR1I3 Q14994 2/20 0.36
PTGES O14684 1/20 0.34
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 2/20 0.33
GAPDH P04406 1/20 0.33
TUBB4A P04350 2/20 0.32
TUBB P07437 2/20 0.32
TUBA3C P0DPH7 2/20 0.32
TUBA1B P68363 2/20 0.32
TUBA4A P68366 2/20 0.32
TUBB4B P68371 2/20 0.32
TUBB3 Q13509 2/20 0.32
TUBB2A Q13885 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27537113 0.86 NPC1 (0.37) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL7680558 0.77 SMN1; SMN2 (0.37) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL7681595 0.77 NR1I3 (0.37) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL7683114 0.75 SMN1; SMN2 (0.38) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL7682758 0.72 CYP11B2 (0.46) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL7676130 0.71 MAPT (0.40) NPC1RAB9ASMN1; SMN2PTGESMAPT
SCHEMBL7678666 0.69 RORC (0.33) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL15958653 0.68 KDM4E (0.49) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL7676206 0.66 HRH4 (0.38) NR1I3PTGESPGK1
SCHEMBL7681496 0.65 SMN1; SMN2 (0.43) SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376490-B1 STRONG N-METHYL-D-ASPARATE RECEPTOR ANTAGONISTS; USEFUL IN TREATING STROKES, ISCHEMIA, AND CENTRAL NERVOUS SYSTEM INJURIES PFIZER INC 2002-04-23 US disclosed
EP-0885212-B1 QUINOXALINEDIONES PFIZER RES AND BR DEV COMPANY (IE) 2001-11-14 EP disclosed