SCHEMBL7675092

SCHEMBL7675092

COC(=O)c1ccc(-c2c(NC(=O)C(F)(F)F)nc3ccc(C(=O)c4ccccc4)cn23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 6/20 0.47
AKT2 P31751 6/20 0.47
ALDH1A1 P00352 5/20 0.43
ALDH1A3 P47895 1/20 0.43
USP7 Q93009 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TNKS O95271 1/20 0.39
PTPN1 P18031 1/20 0.39
CDK2 P24941 2/20 0.39
KDM4E B2RXH2 3/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7673955 0.91 NPC1 (0.42) AKT1AKT2USP7MAPTCDK2
SCHEMBL7676761 0.91 AKT1 (0.51) AKT1AKT2ALDH1A1ALDH1A3USP7
SCHEMBL7679500 0.91 CDK2 (0.43) AKT1AKT2USP7CDK2TRPM8
SCHEMBL7680199 0.89 TLR7 (0.39) AKT1AKT2USP7MAPTCDK2
SCHEMBL7682045 0.89 CDK2 (0.43) AKT1AKT2ALDH1A1USP7MAPT
SCHEMBL7677596 0.88 CDK2 (0.41) AKT1AKT2USP7MAPTNPSR1
SCHEMBL7680034 0.88 CDK2 (0.40) AKT1AKT2USP7MAPTCDK2
SCHEMBL7674349 0.88 TRPV1 (0.40) USP7CDK2CDK4
SCHEMBL7680009 0.85 CDK2 (0.39) AKT1AKT2USP7CDK2RAB9A
SCHEMBL7676765 0.85 POLB (0.46) ALDH1A1MAPTCYP2C9CYP2C19CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed