SCHEMBL7675778

SCHEMBL7675778

CCC(OC(C)=O)c1ccsc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.47
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
PABPC1 P11940 1/20 0.35
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
CYP3A4 P08684 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
LCK P06239 1/20 0.32
FYN P06241 1/20 0.32
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9903752 0.84 ALOX5 (0.43) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL6955956 0.81 MTNR1A (0.42) ALOX5ALDH1A1PABPC1APOBEC3AAPOBEC3G
SCHEMBL9902891 0.81 ALOX5 (0.43) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL14033888 0.79 ALOX5 (0.49) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL5039798 0.78 LMNA (0.46) ALOX5ALDH1A1LMNA
SCHEMBL14528798 0.77 ALOX5 (0.51) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL723114 0.77 ALOX5 (0.51) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL14188736 0.77 ALOX5 (0.43) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9608808 0.75 PABPC1 (0.55) ALDH1A1LMNAPABPC1APOBEC3AAPOBEC3G
SCHEMBL2294116 0.75 PABPC1 (0.55) ALDH1A1LMNAPABPC1APOBEC3AAPOBEC3G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362344-B1 REACTING AN ALDEHYDE WITH ORGANOZINC COMPOUND IN PRESENCE OF CATALYTIC ERYTHRO-B-AMINO ALCOHOL BRISTOL-MYERS SQUIBB PHARMA COMPANY 2002-03-26 US disclosed
US-6187918-B1 CHIRAL AMINOALCOHOL CATALYSTS DUPONT PHARMACEUTICALS COMPANY 2001-02-13 US disclosed