SCHEMBL7680020

SCHEMBL7680020

O=C(c1ccccc1)c1ccc2nc(NC(=O)C(F)(F)F)c(-c3ccc(C(F)(F)F)cc3F)n2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 4/20 0.41
CDK4 P11802 2/20 0.40
ABCC9 O60706 1/20 0.37
ABCC8 Q09428 1/20 0.37
KCNJ11 Q14654 1/20 0.37
KCNJ8 Q15842 1/20 0.37
ADORA3 P0DMS8 4/20 0.36
SRD5A2 P31213 1/20 0.36
MAPT P10636 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
EPHX2 P34913 1/20 0.35
RORC P51449 1/20 0.35
NTRK1 P04629 1/20 0.34
LRRK2 Q5S007 1/20 0.34
MGLL Q99685 1/20 0.34
P2RX1 P51575 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7673981 0.94 VNN1 (0.35) CDK2CDK4ABCC9ABCC8KCNJ11
SCHEMBL7676349 0.91 CDK2 (0.42) CDK2CDK4ABCC9ABCC8KCNJ11
SCHEMBL7676916 0.89 CDK2 (0.44) CDK2CDK4ABCC9ABCC8KCNJ11
SCHEMBL7676510 0.88 CDK2 (0.47) CDK2CDK4ABCC9ABCC8KCNJ11
SCHEMBL7676621 0.86 CDK2 (0.43) CDK2CDK4ABCC9ABCC8KCNJ11
SCHEMBL7674349 0.85 TRPV1 (0.40) CDK2CDK4ADORA3SRD5A2NTRK1
SCHEMBL7676795 0.85 CDK2 (0.39) CDK2CDK4ABCC9ABCC8KCNJ11
SCHEMBL7678672 0.85 CNR2 (0.45) CDK2CDK4ADORA3SRD5A2MAPT
SCHEMBL7676377 0.85 CDK2 (0.42) CDK2CDK4ABCC9ABCC8KCNJ11
SCHEMBL7682053 0.84 CDK2 (0.40) CDK2CDK4ABCC9ABCC8KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed