SCHEMBL7682652

SCHEMBL7682652

O=C1CC(c2ccccc2Cl)Cc2[nH]nc(Nc3ccccc3)c21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.42
TP53 P04637 2/20 0.42
RECQL P46063 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
MAPT P10636 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
USP2 O75604 1/20 0.40
PKM P14618 1/20 0.40
BUB1 O43683 4/20 0.40
DHODH Q02127 1/20 0.39
KDM4E B2RXH2 1/20 0.39
XBP1 P17861 1/20 0.39
MAPK1 P28482 1/20 0.39
LDHA P00338 1/20 0.38
LDHB P07195 1/20 0.38
BRD4 O60885 1/20 0.38
EP300 Q09472 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7682873 0.80 HCAR2 (0.50) HCAR2TP53RECQLSMN1; SMN2MAPT
SCHEMBL7683237 0.79 SMN1; SMN2 (0.48) HCAR2TP53RECQLSMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL7683440 0.78 HCAR2 (0.38) HCAR2LMNA
Hydrochloric Acid SCHEMBL7683434 0.78 HCAR2 (0.38) HCAR2LMNA
SCHEMBL7689472 0.76 LMNA (0.47) HCAR2TP53RECQLSMN1; SMN2MAPT
SCHEMBL7681257 0.74 SMN1; SMN2 (0.45) HCAR2TP53RECQLSMN1; SMN2MAPT
SCHEMBL7689656 0.69 TP53 (0.49) HCAR2TP53RECQLSMN1; SMN2MAPT
SCHEMBL7678959 0.68 SMN1; SMN2 (0.49) HCAR2TP53RECQLSMN1; SMN2MAPT
SCHEMBL7689241 0.66 HCAR2 (0.48) HCAR2TP53SMN1; SMN2MAPTALDH1A1
SCHEMBL7688025 0.66 SMN1; SMN2 (0.53) TP53RECQLSMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed