SCHEMBL7678959

SCHEMBL7678959

Cc1c[nH]c2c1C(=O)CC(c1ccccc1Cl)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.49
HTT P42858 2/20 0.49
RXFP1 Q9HBX9 1/20 0.49
USP2 O75604 1/20 0.49
PKM P14618 1/20 0.49
TP53 P04637 2/20 0.48
RECQL P46063 1/20 0.48
MAPT P10636 1/20 0.47
MAPK1 P28482 2/20 0.43
LDHA P00338 2/20 0.42
LDHB P07195 2/20 0.42
ADRA1A P35348 1/20 0.41
KDM4E B2RXH2 1/20 0.41
XBP1 P17861 1/20 0.41
ERBB2 P04626 1/20 0.39
PIM1 P11309 1/20 0.39
FLT3 P36888 1/20 0.39
MAP4K2 Q12851 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7680997 0.87 HTR2C (0.41) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL7683083 0.84 MAP1LC3B (0.39) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL7688025 0.82 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL7685234 0.80 ALOX15 (0.56) SMN1; SMN2ALDH1A1LMNAHTTTP53
SCHEMBL7689656 0.80 TP53 (0.49) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL7683237 0.77 SMN1; SMN2 (0.48) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL16217087 0.74 LMNA (0.69) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL7681186 0.73 TP53 (0.48) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL7689638 0.73 TP53 (0.48) SMN1; SMN2ALDH1A1LMNAHTTRXFP1
SCHEMBL7689215 0.73 TSHR (0.55) SMN1; SMN2ALDH1A1LMNAHTTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed