SCHEMBL7684819

SCHEMBL7684819

Cc1cc(N2CCSCC2)nc(Nc2c(Br)cc(C(C)C)cc2Br)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 4/20 0.40
SLC2A1 P11166 3/20 0.36
ALDH1A1 P00352 5/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HTT P42858 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
POLB P06746 2/20 0.35
MAPT P10636 3/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPK1 P28482 2/20 0.34
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34
NR4A1 P22736 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
TSHR P16473 2/20 0.34
CRHBP P24387 2/20 0.34
CRHR2 Q13324 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045111 0.82 SLC2A1 (0.40) CRHR1SLC2A1ALDH1A1MEN1KMT2A
SCHEMBL7682687 0.74 CRHR1 (0.62) CRHR1
SCHEMBL7680672 0.72 CRHR1 (0.57) CRHR1ALDH1A1KMT2AHTTMAPT
SCHEMBL3406616 0.65 KDM4E (0.44) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL6981234 0.64 CRHR1 (0.40) CRHR1SLC2A1ALDH1A1MEN1KMT2A
SCHEMBL7678043 0.62 MAPT (0.59) CRHR1ALDH1A1MEN1KMT2APOLB
SCHEMBL20042146 0.62 MAPT (0.65) SLC2A1ALDH1A1MEN1KMT2AHTT
SCHEMBL19476873 0.61 SLC2A1 (0.67) SLC2A1ALDH1A1MEN1KMT2AHTT
SCHEMBL12484199 0.61 MEN1 (0.63) SLC2A1ALDH1A1MEN1KMT2AHTT
SCHEMBL12484612 0.61 MEN1 (0.59) SLC2A1ALDH1A1MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO claimed
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed