SCHEMBL7680672

SCHEMBL7680672

Cc1cc(N2CCOCC2)nc(Nc2ccc(C(C)C)cc2Br)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.57
CRHBP P24387 2/20 0.49
CRHR2 Q13324 2/20 0.49
PKM P14618 1/20 0.49
TSHR P16473 1/20 0.49
PIK3CB P42338 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.46
MAPT P10636 4/20 0.46
TP53 P04637 1/20 0.46
MAPK1 P28482 1/20 0.46
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
KDM4E B2RXH2 1/20 0.41
APAF1 O14727 1/20 0.41
LMNA P02545 1/20 0.41
RET P07949 1/20 0.41
ALDH1A1 P00352 2/20 0.40
IGF1R P08069 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7678043 0.81 MAPT (0.59) CRHR1MAPTTP53KMT2ALMNA
SCHEMBL6984429 0.80 ALDH1A1 (0.39) CRHR1CRHBPCRHR2PKMTSHR
SCHEMBL6981234 0.78 CRHR1 (0.40) CRHR1CRHBPCRHR2PKMTSHR
SCHEMBL7684973 0.73 CRHR1 (1.00) CRHR1
SCHEMBL961117 0.73 CRHBP (0.65) CRHBPCRHR2PKMTSHRPIK3CB
SCHEMBL7684819 0.72 CRHR1 (0.40) CRHR1CRHBPCRHR2PKMTSHR
SCHEMBL14818929 0.71 KMT2A (0.64) CRHBPCRHR2PKMTSHRPIK3CB
SCHEMBL7680556 0.71 MAPT (0.43) CRHR1PKMPIK3CBSMN1; SMN2MAPT
SCHEMBL12486039 0.71 MAPT (0.67) CRHBPCRHR2PKMTSHRPIK3CB
SCHEMBL8208478 0.70 CRHR1 (0.54) CRHR1MAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
CN-1142817-A 1N-alkyl-N-arylpyrimidinamines and derivatives thereof DU PONT MERCK PHARMA (US) 1997-02-12 CN disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed