SCHEMBL7685448

SCHEMBL7685448

CSc1ccc(-c2c(OCC(=O)C(C)(C)C)n[nH]c2-c2ccc(F)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 13/20 0.35
GCGR P47871 4/20 0.35
GSK3B P49841 2/20 0.35
MAPK13 O15264 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
LCK P06239 1/20 0.35
RET P07949 1/20 0.35
ALOX5 P09917 1/20 0.35
PRKACA P17612 1/20 0.35
RPS6KB1 P23443 1/20 0.35
MATK P42679 1/20 0.35
FRK P42685 1/20 0.35
MAPK9 P45984 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CSNK1D P48730 1/20 0.35
GSK3A P49840 1/20 0.35
MAPK12 P53778 1/20 0.35
CSNK1G2 P78368 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6624151 0.86 HAO1 (0.39) MAPK14GCGRGSK3BMAPK13PRKD3
SCHEMBL7542111 0.84 PTGS2 (0.44)
SCHEMBL6623410 0.83 CHRNA7 (0.43) ALOX5CDK2
SCHEMBL7538974 0.80 HAO2 (0.43) ALDH1A1ARHTT
SCHEMBL7671604 0.77 ALDH1A1 (0.35) MAPK14GCGRMAPK13MAPK12MAPK11
SCHEMBL6620206 0.74 PTGS2 (0.44)
SCHEMBL6440359 0.74 ALDH1A1 (0.41) MAPK14GCGRGSK3BMAPK13PRKD3
SCHEMBL6622736 0.73 MAPK14 (0.44) MAPK14GCGRGSK3BMAPK13PRKD3
SCHEMBL6623323 0.73 MAPK14 (0.44) MAPK14GCGRGSK3BMAPK13PRKD3
SCHEMBL8639382 0.71 MAPK14 (0.44) MAPK14GCGRGSK3BMAPK13PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472416-B1 Sulfonylphenylpyrazole compounds useful as COX-2 inhibitors ABBOTT LABORATORIES 2002-10-29 US disclosed