SCHEMBL6624151

SCHEMBL6624151

CSc1ccc(-c2c(OCC(=O)c3ccc(F)cc3)n[nH]c2-c2ccc(F)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 1/20 0.39
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MAPK1 P28482 2/20 0.37
PKM P14618 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37
LMNA P02545 2/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
CNR2 P34972 1/20 0.36
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPK14 Q16539 6/20 0.36
GCGR P47871 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7685448 0.86 MAPK14 (0.35) ALDH1A1MAPK14GCGRMAPK13PRKD3
SCHEMBL6619195 0.83 PTGS2 (0.45)
SCHEMBL6440359 0.74 ALDH1A1 (0.41) MAPK1KDM4EALDH1A1LMNANPC1
SCHEMBL6623323 0.74 MAPK14 (0.44) MAPK14GCGRMAPK13PRKD3MAP4K4
SCHEMBL6622736 0.74 MAPK14 (0.44) MAPK14GCGRMAPK13PRKD3MAP4K4
SCHEMBL8639382 0.72 MAPK14 (0.44) MAPK14GCGRMAPK13PRKD3MAP4K4
SCHEMBL6622652 0.70 PTGS2 (0.41) HPGDPOLB
SCHEMBL7542111 0.70 PTGS2 (0.44)
SCHEMBL6623410 0.69 CHRNA7 (0.43) ALOX5CDK2
SCHEMBL3973566 0.69 PKM (0.41) HAO1MAPK1PKMALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206474-B1 SULFONYLPHENYLPYRAZOLE COMPOUNDS USEFUL AS COX-2 INHIBITORS ABBOTT LAB (US) 2004-05-26 EP disclosed
US-6472416-B1 Sulfonylphenylpyrazole compounds useful as COX-2 inhibitors ABBOTT LABORATORIES 2002-10-29 US disclosed