SCHEMBL7686772

SCHEMBL7686772

CC(C)(C)S(=O)(=O)Nc1ccccc1OBOc1ccccc1NS(=O)(=O)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
NPC1 O15118 1/20 0.38
CA2 P00918 1/20 0.38
ALDH1A1 P00352 5/20 0.37
HTT P42858 1/20 0.37
SLC22A12 Q96S37 2/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
LMNA P02545 1/20 0.35
POLB P06746 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1797703 0.81 KEAP1 (0.49) TSHRALDH1A1SLC22A12PTGS1PTGS2
SCHEMBL9128897 0.78 NPC1 (0.37) TSHRNPC1CA2ALDH1A1HTT
SCHEMBL12932924 0.73 ALDH1A1 (0.50) TSHRNPC1CA2ALDH1A1PTGS1
SCHEMBL14830771 0.72 PSIP1 (0.59) TSHRNPC1CA2ALDH1A1SLC22A12
SCHEMBL5849242 0.72 CA2 (0.46) NPC1CA2HTTMEN1KMT2A
SCHEMBL6880631 0.70 APP (0.44) TSHRNPC1CA2ALDH1A1HTT
SCHEMBL384055 0.70 LMNA (0.56) TSHRALDH1A1KMT2ALMNAPOLB
SCHEMBL3831681 0.69 CA2 (0.40) CA2KMT2A
SCHEMBL20290538 0.69 KMT2A (0.55) TSHRCA2ALDH1A1SLC22A12MEN1
SCHEMBL3066546 0.69 SLC22A12 (0.43) CA2ALDH1A1HTTSLC22A12PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399627-B1 ANTICOAGULANTS; PROTHROMINASE, SERINE PROTEASE INHIBITOR; ACRYLAMIDE DERIVATIVES COR THERAPEUTICS, INC. 2002-06-04 US disclosed
EP-1159264-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2001-12-05 EP disclosed
WO-2000047554-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC. (US) 2000-08-17 WO disclosed