SCHEMBL7687301

SCHEMBL7687301

CCCC1=C(C(=O)SCC)C(C)N=C(c2ccccc2)C1(CC)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 17/20 0.41
TRPV1 Q8NER1 3/20 0.38
GMNN O75496 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
TMIGD3 P0DMS9 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
MAPK1 P28482 1/20 0.35
ADORA2A P29274 1/20 0.35
CYP2C19 P33261 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7678789 0.69 ADORA3 (0.39) ADORA3TRPV1
SCHEMBL7685039 0.62 ADORA3 (0.78) ADORA3TRPV1GMNNCYP1A2CYP3A4
SCHEMBL7461390 0.57 ADORA3 (0.74) ADORA3GMNNCYP1A2CYP3A4TMIGD3
SCHEMBL1641518 0.57 HDAC3 (0.55) CYP3A4TSHRMAPK1MEN1KMT2A
SCHEMBL29742701 0.55 TSHR (0.45) ADORA3CYP3A4TSHRMAPK1
SCHEMBL10174705 0.53 ADORA3 (0.41) ADORA3GMNNCYP1A2CYP3A4TMIGD3
SCHEMBL4576444 0.53 L3MBTL1 (0.66) TSHR
Bicarbonate SCHEMBL27643185 0.52 FFAR1 (0.62) TSHRMEN1GAAKMT2A
Biphenyl SCHEMBL17473044 0.52 THRA (0.48) NPSR1
SCHEMBL19543224 0.52 ALDH1A1 (0.55) MAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376521-B1 ANTIINFLAMMATORY AGENTS; ANTIISCHEMIC AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2002-04-23 US disclosed