SCHEMBL7688235

SCHEMBL7688235

CC1(C)CCC(O)c2cc(N=Nc3ccc(C(=O)O)cc3)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.47
RARG P13631 8/20 0.47
RARA P10276 7/20 0.47
CYP26A1 O43174 2/20 0.47
CYP3A4 P08684 1/20 0.47
CRABP2 P29373 1/20 0.47
RXRA P19793 15/20 0.47
RXRB P28702 12/20 0.47
RXRG P48443 8/20 0.47
MEN1 O00255 1/20 0.43
ABCB11 O95342 1/20 0.43
ESR1 P03372 1/20 0.43
PGR P06401 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD1 P21728 1/20 0.43
TBXA2R P21731 1/20 0.43
SLC6A2 P23975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7688234 1.00 RARB (0.47) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7637331 0.85 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6292739 0.83 RAB9A (0.49) RARBRARGRARAMEN1ESR1
SCHEMBL6292740 0.83 RAB9A (0.49) RARBRARGRARAMEN1ESR1
SCHEMBL6297186 0.81 RXRA (0.42) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6297184 0.81 RXRA (0.42) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8551591 0.81 RXRA (0.66) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8972592 0.81 RXRA (0.66) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8646858 0.79 RXRA (0.41) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6294342 0.78 RARA (0.69) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6465663-B2 ETHYL (E)-4-(2-(5,6-DIHYDRO-5,5-DIMETHYL-NAPHTHALEN-8(7H)-ONE-2 -YL)ETHENYL)BENZOATE AND ETHYL (E)-4-(2-(5,6-DIHYDRO-5,5-DIMETHYL-8-(PHENYLTHIO)-NAPHTHALENYL)ETHENYL) BENZOATE ALLERGAN, INC. 2002-10-15 US disclosed
EP-0915825-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 1999-05-19 EP disclosed
US-5723666-A USEFUL AS REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION ALLERGAN (US) 1998-03-03 US disclosed
WO-1997048672-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1997-12-24 WO disclosed