SCHEMBL7693402

SCHEMBL7693402

Cc1c(-c2ccc(O)cc2)[nH]c2ccc(O)c(CCCCCC(=O)N(C)CCOc3ccc(C(F)(F)F)cc3)c12

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.39
NR1I2 O75469 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
PPARA Q07869 2/20 0.33
BRAF P15056 2/20 0.33
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
MGAT2 Q10469 1/20 0.32
PDE2A O00408 1/20 0.32
P2RY12 Q9H244 1/20 0.32
ESRRG P62508 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027686 0.76 ALDH1A1 (0.39) NR1I2
SCHEMBL9356958 0.73 NR1I2 (0.40) NR1I2
SCHEMBL7694915 0.71 ESR1 (0.54)
SCHEMBL7689050 0.70 BCHE (0.40) BCHEACHE
SCHEMBL7695045 0.69 BCHE (0.37) BCHEACHE
SCHEMBL8789363 0.67 MAPK1 (0.36) NR1I2
SCHEMBL9027574 0.67 DRD2 (0.39)
SCHEMBL8790260 0.66 ESR1 (0.39) NR1I2
SCHEMBL9029036 0.66 TLR9 (0.41)
SCHEMBL7692326 0.66 ESR1 (0.43) NR1I2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002081444-A1 1-INDOLYL DERIVATIVES, USE THEREOF FOR PRODUCTION OF MEDICAMENTS, A METHOD FOR PRODUCTION OF SAID 1-INDOLYL DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING 1-INDOLYL DERIVATIVES SCHERING AKTIENGESELLSCHAFT (DE) 2002-10-17 WO disclosed