SCHEMBL7694273

SCHEMBL7694273

CC1=C(CN2CCCC2)COc2cc(NC(=O)C(Cc3ccccc3)NC(=O)O)ccc21

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.43
ROCK1 Q13464 1/20 0.43
PSMB8 P28062 2/20 0.42
PSMB5 P28074 2/20 0.42
PSMB10 P40306 2/20 0.42
PSMB2 P49721 2/20 0.42
PSMB9 P28065 1/20 0.42
TSHR P16473 1/20 0.40
TRPV1 Q8NER1 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 2/20 0.39
PGR P06401 1/20 0.39
USP30 Q70CQ3 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5582592 0.79 ROCK2 (0.56) ROCK2TSHRTRPV1ALDH1A1HTT
SCHEMBL5582721 0.75 RAB9A (0.55) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL5582928 0.73 CACNA2D1 (0.46) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL5582638 0.72 CYP3A4 (0.53) NPC1RAB9ASMN1; SMN2
SCHEMBL5582758 0.72 USP2 (0.42) ROCK2ROCK1TSHRTRPV1ALDH1A1
SCHEMBL5582749 0.68 ACHE (0.41) KMT2AMEN1ALDH1A1
SCHEMBL18983568 0.65 SMN1; SMN2 (0.56) KMT2AMEN1SMN1; SMN2
SCHEMBL4526386 0.65 FPR2 (0.67) KMT2AMEN1NPC1RAB9ASMN1; SMN2
SCHEMBL6410493 0.65 MMP1 (0.57) PSMB8PSMB5PSMB10PSMB2PSMB9
SCHEMBL6248582 0.64 TACR2 (0.65) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218336-A2 MELANIN CONCENTRATING HORMONE ANTAGONIST Takeda Chemical Industries, Ltd. (JP) 2002-07-03 EP disclosed
WO-2001021577-A2 MELANIN CONCENTRATING HORMONE ANTAGONIST TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-03-29 WO disclosed