SCHEMBL7695

SCHEMBL7695

O=C(O)CN(C(=O)c1cccc([N+](=O)[O-])c1[N+](=O)[O-])c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
LMNA P02545 1/20 0.47
GPR35 Q9HC97 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TSHR P16473 3/20 0.41
CTSD P07339 1/20 0.41
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
TP53 P04637 2/20 0.39
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3134710 0.89 ALDH1A1 (0.57) ALDH1A1LMNASMN1; SMN2TSHRCTSD
SCHEMBL7055735 0.78 CES2 (0.54) ALDH1A1LMNASMN1; SMN2KMT2ACYP1A2
SCHEMBL1418030 0.78 CES2 (0.54) ALDH1A1LMNASMN1; SMN2KMT2ACYP1A2
SCHEMBL30893562 0.75 TSHR (0.68) ALDH1A1GPR35TSHRCTSDKMT2A
SCHEMBL3671 0.75 TSHR (0.68) ALDH1A1GPR35TSHRCTSDKMT2A
SCHEMBL6226801 0.74 GPR35 (0.42) ALDH1A1GPR35TSHRCYP1A2
Potassium Ion SCHEMBL16267317 0.73 TSHR (0.66) ALDH1A1GPR35TSHRCTSDKMT2A
SCHEMBL10824707 0.73 TSHR (0.66) ALDH1A1GPR35TSHRCTSDKMT2A
SCHEMBL16267318 0.73 TSHR (0.66) ALDH1A1GPR35TSHRCTSDKMT2A
SCHEMBL7791983 0.73 TSHR (0.66) ALDH1A1GPR35TSHRCTSDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5091 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3169430-B1 NEW ULTRAHIGH EFFICIENCY, SUPERFICIALLY POROUS PARTICLE (SPP) CHIRAL PHASES FOR LIQUID CHROMATOGRAPHY AZYP LLC (US) 2021-11-10 EP claimed
US-10272364-B2 Superficially porous particle (SPP) chiral phases for liquid chromatography AZYP, LLC (US) 2019-04-30 US claimed
US-20170197156-A1 NEW ULTRAHIGH EFFICIENCY, SUPERFICIALLY POROUS PARTICLE (SPP) CHIRAL PHASES FOR LIQUID CHROMATOGRAPHY AZYP, LLC (US) 2017-07-13 US claimed
EP-3169430-A1 NEW ULTRAHIGH EFFICIENCY, SUPERFICIALLY POROUS PARTICLE (SPP) CHIRAL PHASES FOR LIQUID CHROMATOGRAPHY Azyp LLC (US) 2017-05-24 EP claimed
WO-2016011425-A1 NEW ULTRAHIGH EFFICIENCY, SUPERFICIALLY POROUS PARTICLE (SPP) CHIRAL PHASES FOR LIQUID CHROMATOGRAPHY AZYP, LLC (US) 2016-01-21 WO claimed
EP-1149099-A2 IMIDAZO[4,5-C]-PYRIDINE-4-ON-DERIVATIVES MERCK PATENT GmbH (DE) 2001-10-31 EP claimed
WO-2000040583-A2 IMIDAZO[4,5-C]-PYRIDINE-4-ON-DERIVATIVES MERCK PATENT GMBH (DE) 2000-07-13 WO claimed
US-5786428-A POLYMER MATRIX OF UNSATURATED MONOMER AND METAL COMPLEX HAVING A LIGAND AND A POLYMERIZABLE UNSATURATED MOIETY; EFFICIENT, RAPID AND SIMPLE PURIFICATION; MEDICAL DIAGNOSIS; CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-07-28 US claimed
US-6432953-B1 None US disclosed
CN-122094690-A Pharmaceutical composition comprising Maraglinib (MARALIXIBAT) and use thereof 2026-05-26 CN disclosed
CN-122071439-A Benzo-ring-containing compounds as protein tyrosine phosphatase inhibitors and uses thereof 湖北生物医药产业技术研究院有限公司 2026-05-22 CN disclosed
WO-2026103853-A1 TSHR ANTAGONIST COMPOUND, PHARMACEUTICAL COMPOSITION, METHOD FOR PREPARING SAME, AND USE THEREOF 长春金赛药业有限责任公司 2026-05-21 WO disclosed
WO-2026103887-A1 PROLINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 北京康辰药业股份有限公司 2026-05-21 WO disclosed
CN-122070482-A Methods of using neurofilament light chain immunoassays 美国西门子医学诊断股份有限公司 2026-05-19 CN disclosed
EP-0301402-A1 Leukotriene antagonists, process for their preparation and their use in the treatment of illnesses HOECHST AKTIENGESELLSCHAFT (DE) 1989-02-01 EP disclosed
EP-0299558-A1 Process for the preparation of ibuprofen GIST-BROCADES N.V. (NL) 1989-01-18 EP disclosed
EP-0299559-A1 Process for the preparation of 2-aryloxypropionic acids GIST-BROCADES N.V. (NL) 1989-01-18 EP disclosed
US-4788199-A ANXIOLYTICS, ANTICONVULSANTS, ANTIANGINA AGENTS RHONE-POULENC SANTE (FR) 1988-11-29 US disclosed
US-4788204-A TRANQUILIZERS; ANTICONVULSANTS; ANGINA AND IMMUNODIFICIENCY TREATMENTS RHONE-POULENC SANTE (FR) 1988-11-29 US disclosed
EP-0210084-A1 Amides, processes for their preparation and medicaments containing them RHONE-POULENC SANTE (FR) 1987-01-28 EP disclosed