SCHEMBL7698087

SCHEMBL7698087

CS(=O)(=O)NCC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(Nc2ccc3ccccc3c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.51
CA1 P00915 4/20 0.47
ACE P12821 2/20 0.47
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
CTSS P25774 1/20 0.45
CTSK P43235 1/20 0.45
CA12 O43570 2/20 0.44
CA9 Q16790 2/20 0.44
PTPN1 P18031 2/20 0.43
PIN1 Q13526 2/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.42
RAB9A P51151 1/20 0.42
HPGDS O60760 1/20 0.41
KAT6A Q92794 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703492 0.90 CA2 (0.42) CA2CA1ACECTSLCTSB
SCHEMBL7700700 0.89 CA2 (0.52) CA2CA1ACECTSLCTSB
SCHEMBL7706585 0.89 ALDH1A1 (0.53) CA2CA1CA12CA9MEN1
SCHEMBL7428036 0.85 CA2 (0.45) CA2CA1ACECA12CA9
SCHEMBL7702953 0.84 PTPN1 (0.53) CA2ACECTSLCTSBCTSS
SCHEMBL7701294 0.83 CA2 (0.50) CA2CA1ACECTSLCTSB
SCHEMBL7694179 0.82 AKR1C3 (0.48) CA2ALDH1A1GAAKAT6A
SCHEMBL7701184 0.81 USP30 (0.49) CA2CA1ACECA12CA9
SCHEMBL7694857 0.81 CA2 (0.43) CA2CA1ACECTSLCTSB
SCHEMBL7702126 0.81 PLAT (0.45) CA2CA1KAT6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed