SCHEMBL7702126

SCHEMBL7702126

Cc1cc(Nc2ccc3ccccc3c2)ccc1C(=O)N[C@@H](Cc1ccccc1)C(=O)CNS(=O)(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PLAT P00750 2/20 0.45
PLAU P00749 1/20 0.43
NPY5R Q15761 1/20 0.43
CA2 P00918 3/20 0.43
KAT6A Q92794 2/20 0.42
MMP9 P14780 2/20 0.42
KCNA5 P22460 2/20 0.42
CASP1 P29466 1/20 0.41
F2 P00734 1/20 0.41
POLB P06746 1/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
CCKAR P32238 1/20 0.39
CCKBR P32239 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CA1 P00915 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703492 0.91 CA2 (0.42) PLATCA2CCKARCCKBRL3MBTL1
SCHEMBL7700700 0.89 CA2 (0.52) PLATCA2KAT6AMMP9CASP1
SCHEMBL7421589 0.88 PYGL (0.43) PLATCA2KAT6ACASP1CCKBR
SCHEMBL7703565 0.82 CA2 (0.51) PLATPLAUNPY5RCA2KAT6A
SCHEMBL7698087 0.81 CA2 (0.51) CA2KAT6ACA1
SCHEMBL7701518 0.80 CA2 (0.44) PLATPLAUNPY5RCA2KAT6A
SCHEMBL7683061 0.78 PYGL (0.43) CA2KAT6ACASP1CCKBR
SCHEMBL7684139 0.78 CA2 (0.48) CA2KAT6AF2CCKBRCA1
SCHEMBL7692550 0.77 AKR1C3 (0.51) PLATPLAUCA2KAT6AF2
SCHEMBL7698802 0.77 CAPN1 (0.67) PLATCA2KAT6AKCNA5CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed