SCHEMBL7701294

SCHEMBL7701294

CS(=O)(=O)NCC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(SCc2ccc3ccccc3c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.50
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
ACE P12821 3/20 0.41
CA1 P00915 3/20 0.41
RAB9A P51151 2/20 0.41
PTPN1 P18031 3/20 0.41
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
RECQL P46063 1/20 0.40
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39
PIN1 Q13526 2/20 0.39
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704769 0.90 CA2 (0.52) CA2CTSLCTSBCTSSCTSK
SCHEMBL7682464 0.88 CA2 (0.42) CA2CTSLCTSBCTSSCTSK
SCHEMBL7696723 0.87 CTSS (0.50) CA2CTSLCTSBCTSSCTSK
SCHEMBL7694676 0.87 CTSL (0.49) CA2CTSLCTSBCTSSCTSK
SCHEMBL7702953 0.84 PTPN1 (0.53) CA2CTSLCTSBCTSSCTSK
SCHEMBL7698087 0.83 CA2 (0.51) CA2CTSLCTSBCTSSCTSK
SCHEMBL7686484 0.80 CA2 (0.44) CA2CTSLCTSBCTSSCTSK
SCHEMBL7706585 0.80 ALDH1A1 (0.53) CA2CA1GAACA12CA9
SCHEMBL7694857 0.78 CA2 (0.43) CA2CTSLCTSBCTSSCTSK
SCHEMBL7661370 0.76 CCKBR (0.44) CA2CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed