SCHEMBL7700170

SCHEMBL7700170

Cn1nc(CC(N)=O)cc1C1=NCCc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 2/20 0.37
MAOA P21397 3/20 0.35
PKM P14618 1/20 0.34
RAD52 P43351 1/20 0.34
PLA2G10 O15496 2/20 0.33
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32
MCTS1 Q9ULC4 1/20 0.32
BCAT2 O15382 1/20 0.32
NOTUM Q6P988 1/20 0.32
MAPT P10636 3/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705891 0.89 ALDH1A1 (0.38) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL7703215 0.80 KMT2A (0.44) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL7702368 0.77 NOS3 (0.41) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL7698346 0.76 TSHR (0.42) ALDH1A1MAPTNPSR1MEN1KMT2A
SCHEMBL5213961 0.71 ALDH1A1 (0.55) NOS3NOS2ALDH1A1KDM4EMAOA
Hydrochloric Acid SCHEMBL8331052 0.70 ALDH1A1 (0.54) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL8510510 0.67 NOS3 (0.41) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL28842917 0.66 PARP1 (0.43) KDM4EPLA2G10BCAT2
SCHEMBL7702576 0.66 PRCP (0.43) MAPTNPSR1MEN1KMT2A
SCHEMBL7706815 0.65 BCAT2 (0.47) NOS3NOS2ALDH1A1KDM4EMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed