SCHEMBL7698452

SCHEMBL7698452

COc1ccc(N)c(C(=O)NC(=O)CN)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.48
RAF1 P04049 1/20 0.46
ARAF P10398 1/20 0.46
BRAF P15056 1/20 0.46
HDAC1 Q13547 1/20 0.46
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 5/20 0.44
HPGD P15428 2/20 0.44
TSHR P16473 2/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
ADRA1A P35348 1/20 0.44
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
RAB9A P51151 1/20 0.41
KLKB1 P03952 1/20 0.41
GAA P10253 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199077 0.83 BRAF (0.51) NOS2RAF1ARAFBRAFHDAC1
SCHEMBL6394247 0.80 BRAF (0.51) NOS2RAF1ARAFBRAFHDAC1
SCHEMBL1558756 0.80 BRAF (0.65) NOS2RAF1ARAFBRAFHDAC1
SCHEMBL13753817 0.79 HPGD (0.52) NOS2RAF1ARAFBRAFHDAC1
SCHEMBL7698671 0.77 KEAP1 (0.54) BRAFHDAC1ALDH1A1
SCHEMBL11026476 0.77 NOS2 (0.62) NOS2RAF1ARAFBRAFHDAC1
SCHEMBL267307 0.76 KDM4E (0.62) NOS2KDM4EALDH1A1HPGDTSHR
SCHEMBL7698207 0.76 ERAP2 (0.46) NOS2
SCHEMBL13958731 0.76 ALDH1A1 (0.49) NOS2RAF1ARAFBRAFHDAC1
Hydrochloric Acid SCHEMBL5100210 0.74 ALDH1A1 (0.60) NOS2KDM4EALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002028829-A2 PEPTIDE DEFORMYLASE INHIBITORS QUESTCOR PHARMACEUTICALS, INC. (US) 2002-04-11 WO claimed