SCHEMBL7698671

SCHEMBL7698671

NCC(=O)NC(=O)c1cc(F)ccc1N

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.54
FADS1 O60427 1/20 0.49
HDAC1 Q13547 9/20 0.40
PYGL P06737 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
HDAC3 O15379 3/20 0.38
ALDH1A1 P00352 1/20 0.37
BRAF P15056 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36
HDAC2 Q92769 2/20 0.35
GCK P35557 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24210299 0.81 KEAP1 (0.63) KEAP1FADS1HDAC1CES2CES1
SCHEMBL7698452 0.77 NOS2 (0.48) HDAC1ALDH1A1BRAF
SCHEMBL1559256 0.77 KEAP1 (0.58) KEAP1FADS1HDAC1CES2CES1
SCHEMBL690577 0.76 KEAP1 (0.61) KEAP1FADS1HDAC1CES2CES1
SCHEMBL29520286 0.75 KEAP1 (0.56) KEAP1FADS1HDAC1CES2CES1
SCHEMBL13753884 0.75 KEAP1 (0.56) KEAP1FADS1HDAC1CES2CES1
SCHEMBL15630978 0.74 KEAP1 (0.59) KEAP1FADS1HDAC1HDAC3HDAC2
SCHEMBL11575893 0.73 KEAP1 (0.58) KEAP1FADS1HDAC1CES2CES1
SCHEMBL4333053 0.72 KEAP1 (0.56) KEAP1FADS1HDAC1ALDH1A1BRAF
SCHEMBL135091 0.71 KEAP1 (1.00) KEAP1FADS1HDAC1PYGLCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002028829-A2 PEPTIDE DEFORMYLASE INHIBITORS QUESTCOR PHARMACEUTICALS, INC. (US) 2002-04-11 WO claimed