SCHEMBL7698563

SCHEMBL7698563

O=C(O)Nc1cc(COC2CCCCO2)c(I)cc1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 4/20 0.40
CREBBP Q92793 2/20 0.38
ALDH1A1 P00352 6/20 0.38
MAPT P10636 5/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 6/20 0.36
MEN1 O00255 4/20 0.35
HPGD P15428 2/20 0.35
EP300 Q09472 1/20 0.34
KDM4E B2RXH2 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
GSTP1 P09211 1/20 0.34
GSTM2 P28161 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7140551 0.89 HCAR3 (0.36) HCAR3CREBBPALDH1A1MAPTL3MBTL1
SCHEMBL7703580 0.82 HCAR3 (0.38) HCAR3CREBBPALDH1A1MAPTL3MBTL1
SCHEMBL7700574 0.82 ALDH1A1 (0.38) HCAR3CREBBPALDH1A1MAPTL3MBTL1
SCHEMBL5563454 0.76 KMT2A (0.38) HCAR3CREBBPALDH1A1MAPTL3MBTL1
SCHEMBL7143475 0.73 KMT2A (0.35) HCAR3CREBBPALDH1A1MAPTL3MBTL1
SCHEMBL7147995 0.73 ALDH1A1 (0.36) HCAR3CREBBPALDH1A1MAPTL3MBTL1
SCHEMBL7139585 0.72 MMP8 (0.35) HCAR3CREBBPALDH1A1MAPTL3MBTL1
SCHEMBL20985428 0.72 HCAR3 (0.49) HCAR3ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL20985427 0.72 HCAR3 (0.49) HCAR3ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL7139514 0.72 CHRM3 (0.35) HCAR3CREBBPALDH1A1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed